Siponimod: Disentangling disability and relapses in secondary progressive multiple sclerosis

In multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses. To distinguish siponimod's direct effects on disability progression from those on relapses in the EXPAND phase 3 trial. Three estimands, one based on principal stratum and...

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Published in:Multiple sclerosis Vol. 27; no. 10; p. 1564
Main Authors: Cree, Bruce Ac, Magnusson, Baldur, Rouyrre, Nicolas, Fox, Robert J, Giovannoni, Gavin, Vermersch, Patrick, Bar-Or, Amit, Gold, Ralf, Piani Meier, Daniela, Karlsson, Göril, Tomic, Davorka, Wolf, Christian, Dahlke, Frank, Kappos, Ludwig
Format: Journal Article
Language:English
Published: England 01.09.2021
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ISSN:1477-0970, 1477-0970
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Abstract In multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses. To distinguish siponimod's direct effects on disability progression from those on relapses in the EXPAND phase 3 trial. Three estimands, one based on principal stratum and two on hypothetical scenarios (no relapses, or equal relapses in both treatment arms), were defined to determine the extent to which siponimod's effects on 3- and 6-month confirmed disability progression were independent of on-study relapses. Principal stratum analysis estimated that siponimod reduced the risk of 3- and 6-month confirmed disability progression by 14%-20% and 29%-33%, respectively, compared with placebo in non-relapsing patients. In the hypothetical scenarios, risk reductions independent of relapses were 14%-18% and 23% for 3- and 6-month confirmed disability progression, respectively. By controlling the confounding impact of on-study relapses on confirmed disability progression, these statistical approaches provide a methodological framework to assess treatment effects on disability progression in relapsing and non-relapsing patients. The analyses support that siponimod may be useful for treating secondary progressive multiple sclerosis in patients with or without relapses.
AbstractList In multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses. To distinguish siponimod's direct effects on disability progression from those on relapses in the EXPAND phase 3 trial. Three estimands, one based on principal stratum and two on hypothetical scenarios (no relapses, or equal relapses in both treatment arms), were defined to determine the extent to which siponimod's effects on 3- and 6-month confirmed disability progression were independent of on-study relapses. Principal stratum analysis estimated that siponimod reduced the risk of 3- and 6-month confirmed disability progression by 14%-20% and 29%-33%, respectively, compared with placebo in non-relapsing patients. In the hypothetical scenarios, risk reductions independent of relapses were 14%-18% and 23% for 3- and 6-month confirmed disability progression, respectively. By controlling the confounding impact of on-study relapses on confirmed disability progression, these statistical approaches provide a methodological framework to assess treatment effects on disability progression in relapsing and non-relapsing patients. The analyses support that siponimod may be useful for treating secondary progressive multiple sclerosis in patients with or without relapses.
In multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses.BACKGROUNDIn multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses.To distinguish siponimod's direct effects on disability progression from those on relapses in the EXPAND phase 3 trial.OBJECTIVETo distinguish siponimod's direct effects on disability progression from those on relapses in the EXPAND phase 3 trial.Three estimands, one based on principal stratum and two on hypothetical scenarios (no relapses, or equal relapses in both treatment arms), were defined to determine the extent to which siponimod's effects on 3- and 6-month confirmed disability progression were independent of on-study relapses.METHODSThree estimands, one based on principal stratum and two on hypothetical scenarios (no relapses, or equal relapses in both treatment arms), were defined to determine the extent to which siponimod's effects on 3- and 6-month confirmed disability progression were independent of on-study relapses.Principal stratum analysis estimated that siponimod reduced the risk of 3- and 6-month confirmed disability progression by 14%-20% and 29%-33%, respectively, compared with placebo in non-relapsing patients. In the hypothetical scenarios, risk reductions independent of relapses were 14%-18% and 23% for 3- and 6-month confirmed disability progression, respectively.RESULTSPrincipal stratum analysis estimated that siponimod reduced the risk of 3- and 6-month confirmed disability progression by 14%-20% and 29%-33%, respectively, compared with placebo in non-relapsing patients. In the hypothetical scenarios, risk reductions independent of relapses were 14%-18% and 23% for 3- and 6-month confirmed disability progression, respectively.By controlling the confounding impact of on-study relapses on confirmed disability progression, these statistical approaches provide a methodological framework to assess treatment effects on disability progression in relapsing and non-relapsing patients. The analyses support that siponimod may be useful for treating secondary progressive multiple sclerosis in patients with or without relapses.CONCLUSIONBy controlling the confounding impact of on-study relapses on confirmed disability progression, these statistical approaches provide a methodological framework to assess treatment effects on disability progression in relapsing and non-relapsing patients. The analyses support that siponimod may be useful for treating secondary progressive multiple sclerosis in patients with or without relapses.
Author Magnusson, Baldur
Fox, Robert J
Cree, Bruce Ac
Bar-Or, Amit
Vermersch, Patrick
Tomic, Davorka
Rouyrre, Nicolas
Karlsson, Göril
Gold, Ralf
Dahlke, Frank
Piani Meier, Daniela
Kappos, Ludwig
Giovannoni, Gavin
Wolf, Christian
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  organization: Novartis Pharma AG, Basel, Switzerland
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  organization: Novartis Pharma AG, Basel, Switzerland
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  orcidid: 0000-0002-4263-3717
  surname: Fox
  fullname: Fox, Robert J
  organization: Mellen Center for Multiple Sclerosis Treatment and Research, Neurological Institute, Cleveland Clinic, Cleveland, OH, USA
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  organization: Blizard Institute, Barts and The London School of Medicine and Dentistry, Queen Mary University of London, London, UK
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  surname: Bar-Or
  fullname: Bar-Or, Amit
  organization: Center for Neuroinflammation and Experimental Therapeutics and Multiple Sclerosis Division, Department of Neurology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, PA, USA/Neuroimmunology Unit, Montreal Neurological Institute and Hospital, McGill University, Montreal, QC, Canada
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  fullname: Gold, Ralf
  organization: Department of Neurology, St. Josef-Hospital, Ruhr-University Bochum, Bochum, Germany
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  organization: Novartis Pharma AG, Basel, Switzerland
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  organization: Novartis Pharma AG, Basel, Switzerland
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  orcidid: 0000-0002-4683-0507
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  surname: Kappos
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  organization: Neurologic Clinic and Policlinic, Departments of Medicine, Clinical Research, Biomedicine and Biomedical Engineering, University Hospital, University of Basel, Basel, Switzerland
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Multiple sclerosis
relapses
secondary progressive multiple sclerosis
progressive multiple sclerosis
siponimod
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Snippet In multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses. To distinguish siponimod's direct...
In multiple sclerosis, impact of treatment on disability progression can be confounded if treatment also reduces relapses.BACKGROUNDIn multiple sclerosis,...
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SubjectTerms Azetidines - therapeutic use
Benzyl Compounds - therapeutic use
Disease Progression
Humans
Multiple Sclerosis, Chronic Progressive - drug therapy
Recurrence
Title Siponimod: Disentangling disability and relapses in secondary progressive multiple sclerosis
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