The Nucleotide-Free State of the Cannabinoid CB2/Gi Complex
In this issue of Cell, two papers report agonist-bound cryo-EM structures of the cannabinoid receptor, CB2, in complex with Gi. Importantly, beyond providing information that could help distinguish CB2 ligand binding from CB1, these structures support the existence of a nucleotide-free state during...
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| Veröffentlicht in: | Cell Jg. 180; H. 4; S. 603 |
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| Sprache: | Englisch |
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20.02.2020
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| ISSN: | 1097-4172, 1097-4172 |
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| Abstract | In this issue of Cell, two papers report agonist-bound cryo-EM structures of the cannabinoid receptor, CB2, in complex with Gi. Importantly, beyond providing information that could help distinguish CB2 ligand binding from CB1, these structures support the existence of a nucleotide-free state during G-protein signaling. |
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| AbstractList | In this issue of Cell, two papers report agonist-bound cryo-EM structures of the cannabinoid receptor, CB2, in complex with Gi. Importantly, beyond providing information that could help distinguish CB2 ligand binding from CB1, these structures support the existence of a nucleotide-free state during G-protein signaling. In this issue of Cell, two papers report agonist-bound cryo-EM structures of the cannabinoid receptor, CB2, in complex with Gi. Importantly, beyond providing information that could help distinguish CB2 ligand binding from CB1, these structures support the existence of a nucleotide-free state during G-protein signaling.In this issue of Cell, two papers report agonist-bound cryo-EM structures of the cannabinoid receptor, CB2, in complex with Gi. Importantly, beyond providing information that could help distinguish CB2 ligand binding from CB1, these structures support the existence of a nucleotide-free state during G-protein signaling. |
| Author | Hurst, Dow P Reggio, Patricia H Lynch, Diane L |
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| BackLink | https://www.ncbi.nlm.nih.gov/pubmed/32084338$$D View this record in MEDLINE/PubMed |
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| Title | The Nucleotide-Free State of the Cannabinoid CB2/Gi Complex |
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