Suchergebnisse - "Enfuvirtide"
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1
Autoren: et al.
Quelle: Journal of controlled release : official journal of the Controlled Release Society [J Control Release] 2025 Sep 10; Vol. 385, pp. 113954. Date of Electronic Publication: 2025 Jun 16.
Publikationsart: Journal Article
Info zur Zeitschrift: Publisher: Elsevier Science Publishers Country of Publication: Netherlands NLM ID: 8607908 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-4995 (Electronic) Linking ISSN: 01683659 NLM ISO Abbreviation: J Control Release Subsets: MEDLINE
MeSH-Schlagworte: Enfuvirtide*/administration & dosage , Enfuvirtide*/pharmacokinetics , HIV Fusion Inhibitors*/administration & dosage , HIV Fusion Inhibitors*/pharmacokinetics , Drug Delivery Systems*/instrumentation , HIV Envelope Protein gp41*/administration & dosage , HIV Envelope Protein gp41*/pharmacokinetics, Animals ; Rats, Sprague-Dawley ; Administration, Cutaneous ; Needles ; Male ; Polyesters/chemistry ; Skin/metabolism ; Rats ; Povidone/chemistry ; Silicon Dioxide/chemistry ; Microinjections ; Drug Liberation
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2
Autoren: et al.
Quelle: ACS applied materials & interfaces [ACS Appl Mater Interfaces] 2025 May 07; Vol. 17 (18), pp. 26227-26251. Date of Electronic Publication: 2025 Mar 10.
Publikationsart: Journal Article
Info zur Zeitschrift: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101504991 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1944-8252 (Electronic) Linking ISSN: 19448244 NLM ISO Abbreviation: ACS Appl Mater Interfaces Subsets: MEDLINE
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3
Autoren: et al.
Quelle: Journal of virology [J Virol] 2025 May 20; Vol. 99 (5), pp. e0228924. Date of Electronic Publication: 2025 Apr 10.
Publikationsart: Journal Article; Review
Info zur Zeitschrift: Publisher: American Society For Microbiology Country of Publication: United States NLM ID: 0113724 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1098-5514 (Electronic) Linking ISSN: 0022538X NLM ISO Abbreviation: J Virol Subsets: MEDLINE
MeSH-Schlagworte: HIV-1*/drug effects , HIV Fusion Inhibitors*/pharmacology , HIV Fusion Inhibitors*/chemistry , HIV Fusion Inhibitors*/therapeutic use , Drug Discovery*/methods, Humans ; Enfuvirtide ; HIV Envelope Protein gp41/chemistry ; HIV Envelope Protein gp41/pharmacology ; Drug Resistance, Viral ; HIV Infections/drug therapy ; HIV Infections/virology ; Antiviral Agents/pharmacology ; Virus Replication/drug effects
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4
Autoren: et al.
Quelle: European journal of medicinal chemistry [Eur J Med Chem] 2025 Jan 05; Vol. 281, pp. 117017. Date of Electronic Publication: 2024 Nov 01.
Publikationsart: Journal Article; Review
Info zur Zeitschrift: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
MeSH-Schlagworte: Antiviral Agents*/pharmacology , Antiviral Agents*/chemistry , Antiviral Agents*/chemical synthesis , Drug Discovery* , Indoles*/chemistry , Indoles*/pharmacology , Indoles*/chemical synthesis, Animals ; Humans ; Enfuvirtide/chemistry ; Enfuvirtide/pharmacology ; Molecular Structure ; SARS-CoV-2/drug effects ; Structure-Activity Relationship ; Virus Diseases/drug therapy ; Zika Virus/drug effects
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5
Autoren: et al.
Quelle: Journal of biomolecular structure & dynamics [J Biomol Struct Dyn] 2022 Aug; Vol. 40 (12), pp. 5566-5576. Date of Electronic Publication: 2021 Jan 13.
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Taylor & Francis Country of Publication: England NLM ID: 8404176 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1538-0254 (Electronic) Linking ISSN: 07391102 NLM ISO Abbreviation: J Biomol Struct Dyn Subsets: MEDLINE
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6
Autoren: et al.
Quelle: European journal of medicinal chemistry [Eur J Med Chem] 2024 Apr 05; Vol. 269, pp. 116299. Date of Electronic Publication: 2024 Mar 08.
Publikationsart: Journal Article
Info zur Zeitschrift: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
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7
Autoren: et al.
Quelle: Protein and peptide letters [Protein Pept Lett] 2024; Vol. 31 (6), pp. 447-457.
Publikationsart: Journal Article
Info zur Zeitschrift: Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 9441434 Publication Model: Print Cited Medium: Internet ISSN: 1875-5305 (Electronic) Linking ISSN: 09298665 NLM ISO Abbreviation: Protein Pept Lett Subsets: MEDLINE
MeSH-Schlagworte: HIV-1*/drug effects , Drug Design*, Humans ; HIV Fusion Inhibitors/pharmacology ; HIV Fusion Inhibitors/chemistry ; HIV Envelope Protein gp41/chemistry ; HIV Envelope Protein gp41/antagonists & inhibitors ; HIV Envelope Protein gp41/metabolism ; Peptides/chemistry ; Peptides/pharmacology ; Anti-HIV Agents/pharmacology ; Anti-HIV Agents/chemistry ; Enfuvirtide/pharmacology ; Enfuvirtide/chemistry ; Amino Acid Sequence
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8
Autoren: et al.
Quelle: Journal of immunotoxicology [J Immunotoxicol] 2020 Dec; Vol. 17 (1), pp. 59-66.
Publikationsart: Journal Article
Info zur Zeitschrift: Publisher: Informa Healthcare Country of Publication: England NLM ID: 101201960 Publication Model: Print Cited Medium: Internet ISSN: 1547-6901 (Electronic) Linking ISSN: 1547691X NLM ISO Abbreviation: J Immunotoxicol Subsets: MEDLINE
MeSH-Schlagworte: Antibodies, Monoclonal, Humanized/*immunology , Antigen-Presenting Cells/*immunology , Enfuvirtide/*immunology , Glatiramer Acetate/*immunology , Injection Site Reaction/*immunology, Antibodies, Monoclonal, Humanized/administration & dosage ; Antigen Presentation/drug effects ; Antigen-Presenting Cells/drug effects ; Antigen-Presenting Cells/metabolism ; Cytokines/metabolism ; Drug Evaluation, Preclinical/methods ; Enfuvirtide/administration & dosage ; Glatiramer Acetate/administration & dosage ; Humans ; Injections, Subcutaneous/adverse effects ; THP-1 Cells
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9
Autoren: et al.
Quelle: European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V [Eur J Pharm Biopharm] 2019 Apr; Vol. 137, pp. 218-226. Date of Electronic Publication: 2019 Mar 06.
Publikationsart: Comparative Study; Journal Article
Info zur Zeitschrift: Publisher: Elsevier Science Country of Publication: Netherlands NLM ID: 9109778 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-3441 (Electronic) Linking ISSN: 09396411 NLM ISO Abbreviation: Eur J Pharm Biopharm Subsets: MEDLINE
MeSH-Schlagworte: Enfuvirtide/*administration & dosage , HIV/*drug effects , HIV Fusion Inhibitors/*administration & dosage , Polyethylene Glycols/*chemistry, Animals ; Cell Line ; Enfuvirtide/pharmacokinetics ; Enfuvirtide/pharmacology ; Enzyme-Linked Immunosorbent Assay ; HIV Fusion Inhibitors/pharmacokinetics ; HIV Fusion Inhibitors/pharmacology ; HIV Infections/drug therapy ; Humans ; Lymph/metabolism ; Male ; Rats ; Rats, Sprague-Dawley
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10
Autoren: et al.
Quelle: Drug delivery and translational research [Drug Deliv Transl Res] 2023 Aug; Vol. 13 (8), pp. 2183-2193. Date of Electronic Publication: 2023 Apr 29.
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Springer Country of Publication: United States NLM ID: 101540061 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2190-3948 (Electronic) Linking ISSN: 2190393X NLM ISO Abbreviation: Drug Deliv Transl Res Subsets: MEDLINE
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11
Autoren:
Quelle: AIDS research and human retroviruses [AIDS Res Hum Retroviruses] 2019 Oct; Vol. 35 (10), pp. 941-947. Date of Electronic Publication: 2019 Aug 12.
Publikationsart: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Mary Ann Liebert Country of Publication: United States NLM ID: 8709376 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1931-8405 (Electronic) Linking ISSN: 08892229 NLM ISO Abbreviation: AIDS Res Hum Retroviruses Subsets: MEDLINE
MeSH-Schlagworte: Drug Resistance, Viral*/genetics , Mutation* , Software*, DNA Mutational Analysis/*methods , DNA, Viral/*genetics , Enfuvirtide/*pharmacokinetics , HIV Envelope Protein gp41/*genetics , HIV Fusion Inhibitors/*pharmacology , HIV Infections/*drug therapy , HIV-1/*drug effects, Amino Acid Sequence ; Amino Acid Substitution ; Base Sequence ; Databases, Genetic ; Enfuvirtide/therapeutic use ; Global Health ; HIV Envelope Protein gp41/physiology ; HIV Fusion Inhibitors/therapeutic use ; HIV Infections/virology ; HIV-1/classification ; HIV-1/genetics ; HIV-1/isolation & purification ; Humans ; Internet ; Mutation, Missense ; Sequence Alignment ; Sequence Homology, Nucleic Acid
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12
Autoren: et al.
Quelle: AIDS (London, England) [AIDS] 2019 Aug 01; Vol. 33 (10), pp. 1545-1555.
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Lippincott Williams & Wilkins Country of Publication: England NLM ID: 8710219 Publication Model: Print Cited Medium: Internet ISSN: 1473-5571 (Electronic) Linking ISSN: 02699370 NLM ISO Abbreviation: AIDS Subsets: MEDLINE
MeSH-Schlagworte: Drug Discovery/*methods , Enfuvirtide/*chemistry , Enfuvirtide/*pharmacology , HIV Envelope Protein gp41/*chemistry , HIV Envelope Protein gp41/*metabolism , HIV Fusion Inhibitors/*chemistry , HIV Fusion Inhibitors/*pharmacology, Animals ; Binding Sites ; Cell Fusion ; Cell Line ; Enfuvirtide/chemical synthesis ; HIV Core Protein p24/metabolism ; HIV Fusion Inhibitors/chemical synthesis ; Humans ; Protein Binding ; Recombinant Proteins/chemistry ; Recombinant Proteins/metabolism ; Temperature
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13
Autoren: et al.
Quelle: PloS one [PLoS One] 2019 May 23; Vol. 14 (5), pp. e0216712. Date of Electronic Publication: 2019 May 23 (Print Publication: 2019).
Publikationsart: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Public Library of Science Country of Publication: United States NLM ID: 101285081 Publication Model: eCollection Cited Medium: Internet ISSN: 1932-6203 (Electronic) Linking ISSN: 19326203 NLM ISO Abbreviation: PLoS One Subsets: MEDLINE
MeSH-Schlagworte: Enfuvirtide/*pharmacology , Raltegravir Potassium/*pharmacology, Adult ; Alanine Transaminase/analysis ; Alanine Transaminase/blood ; Anti-Retroviral Agents/therapeutic use ; Creatine/analysis ; Creatine/blood ; Enfuvirtide/metabolism ; Enfuvirtide/toxicity ; HIV Infections/drug therapy ; Healthy Volunteers ; Humans ; Insulin Resistance ; Kidney/drug effects ; Leukocytes, Mononuclear/metabolism ; Lipids/analysis ; Liver/drug effects ; Male ; Metabolism/drug effects ; Mitochondria/drug effects ; Raltegravir Potassium/metabolism ; Raltegravir Potassium/toxicity
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14
Autoren: et al.
Quelle: Journal of virology [J Virol] 2019 Dec 12; Vol. 94 (1). Date of Electronic Publication: 2019 Dec 12 (Print Publication: 2019).
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: American Society For Microbiology Country of Publication: United States NLM ID: 0113724 Publication Model: Electronic-Print Cited Medium: Internet ISSN: 1098-5514 (Electronic) Linking ISSN: 0022538X NLM ISO Abbreviation: J Virol Subsets: MEDLINE
MeSH-Schlagworte: Enfuvirtide/*metabolism , HIV Envelope Protein gp41/*chemistry , HIV Fusion Inhibitors/*metabolism , HIV-1/*chemistry , Tryptophan/*chemistry, Amino Acid Motifs ; Binding Sites ; Circular Dichroism ; Enfuvirtide/chemical synthesis ; HEK293 Cells ; HIV Envelope Protein gp41/antagonists & inhibitors ; HIV Envelope Protein gp41/metabolism ; HIV Fusion Inhibitors/chemical synthesis ; HIV-1/metabolism ; Humans ; Protein Binding ; Protein Interaction Domains and Motifs ; Protein Structure, Secondary ; Structure-Activity Relationship ; Tryptophan/metabolism
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15
Autoren: et al.
Quelle: Protein science : a publication of the Protein Society [Protein Sci] 2019 Aug; Vol. 28 (8), pp. 1501-1512.
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Cold Spring Harbor Laboratory Press Country of Publication: United States NLM ID: 9211750 Publication Model: Print Cited Medium: Internet ISSN: 1469-896X (Electronic) Linking ISSN: 09618368 NLM ISO Abbreviation: Protein Sci Subsets: MEDLINE
MeSH-Schlagworte: Peptide Library*, Enfuvirtide/*pharmacology , HIV Envelope Protein gp41/*antagonists & inhibitors , HIV Fusion Inhibitors/*pharmacology, Enfuvirtide/chemistry ; HIV Envelope Protein gp41/chemistry ; HIV Envelope Protein gp41/metabolism ; HIV Fusion Inhibitors/chemistry ; Humans ; Hydrophobic and Hydrophilic Interactions ; Models, Molecular ; Protein Conformation
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16
Autoren: et al.
Quelle: PLoS pathogens [PLoS Pathog] 2019 Feb 04; Vol. 15 (2), pp. e1007552. Date of Electronic Publication: 2019 Feb 04 (Print Publication: 2019).
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Public Library of Science Country of Publication: United States NLM ID: 101238921 Publication Model: eCollection Cited Medium: Internet ISSN: 1553-7374 (Electronic) Linking ISSN: 15537366 NLM ISO Abbreviation: PLoS Pathog Subsets: MEDLINE
MeSH-Schlagworte: Enfuvirtide/*therapeutic use , Lipopeptides/*therapeutic use , Simian Acquired Immunodeficiency Syndrome/*therapy, Animals ; Anti-Retroviral Agents ; Antibodies, Neutralizing ; Drug Resistance, Viral ; Enfuvirtide/pharmacology ; HEK293 Cells ; HIV Fusion Inhibitors/pharmacology ; HIV Fusion Inhibitors/therapeutic use ; HIV Infections/therapy ; HIV-1/pathogenicity ; Humans ; Macaca mulatta/immunology ; Macaca mulatta/metabolism ; Male ; Rats ; Rats, Sprague-Dawley ; Simian Immunodeficiency Virus/pathogenicity ; Viral Load ; Virus Internalization
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17
Autoren: et al.
Quelle: The Journal of biological chemistry [J Biol Chem] 2018 Apr 06; Vol. 293 (14), pp. 5323-5334. Date of Electronic Publication: 2018 Feb 07.
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Elsevier Inc. on behalf of American Society for Biochemistry and Molecular Biology Country of Publication: United States NLM ID: 2985121R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1083-351X (Electronic) Linking ISSN: 00219258 NLM ISO Abbreviation: J Biol Chem Subsets: MEDLINE
MeSH-Schlagworte: Enfuvirtide/*analogs & derivatives , Enfuvirtide/*chemistry , HIV Fusion Inhibitors/*chemistry, Amino Acid Sequence ; Anti-Retroviral Agents/pharmacology ; Crystallography, X-Ray/methods ; Drug Design ; Drug Resistance, Viral/drug effects ; Enfuvirtide/pharmacology ; HIV-1/metabolism ; HIV-1/physiology ; HIV-2/metabolism ; HIV-2/physiology ; Humans ; Lipopeptides/pharmacology ; Peptide Fragments/pharmacology ; Virus Internalization/drug effects
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18
Autoren: et al.
Quelle: PloS one [PLoS One] 2023 Jun 08; Vol. 18 (6), pp. e0286752. Date of Electronic Publication: 2023 Jun 08 (Print Publication: 2023).
Publikationsart: Journal Article; Research Support, Non-U.S. Gov't
Info zur Zeitschrift: Publisher: Public Library of Science Country of Publication: United States NLM ID: 101285081 Publication Model: eCollection Cited Medium: Internet ISSN: 1932-6203 (Electronic) Linking ISSN: 19326203 NLM ISO Abbreviation: PLoS One Subsets: MEDLINE
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19
Autoren: et al.
Quelle: Einstein (Sao Paulo, Brazil) [Einstein (Sao Paulo)] 2023 Apr 17; Vol. 21, pp. eAO0230. Date of Electronic Publication: 2023 Apr 17 (Print Publication: 2023).
Publikationsart: Journal Article
Info zur Zeitschrift: Publisher: Instituto de Ensino e Pesquisa Albert Einstein Country of Publication: Brazil NLM ID: 101281800 Publication Model: eCollection Cited Medium: Internet ISSN: 2317-6385 (Electronic) Linking ISSN: 16794508 NLM ISO Abbreviation: Einstein (Sao Paulo) Subsets: MEDLINE
MeSH-Schlagworte: Rodentia* , Cesarean Section*, Animals ; Rats ; Pregnancy ; Female ; Enfuvirtide ; Rats, Wistar ; Biological Assay
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20
Autoren:
Quelle: Current pharmaceutical biotechnology [Curr Pharm Biotechnol] 2023; Vol. 24 (14), pp. 1774-1783.
Publikationsart: Review; Journal Article
Info zur Zeitschrift: Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 100960530 Publication Model: Print Cited Medium: Internet ISSN: 1873-4316 (Electronic) Linking ISSN: 13892010 NLM ISO Abbreviation: Curr Pharm Biotechnol Subsets: MEDLINE
MeSH-Schlagworte: Virus Diseases*/drug therapy , Viruses*, Humans ; Antiviral Agents/pharmacology ; Antiviral Agents/therapeutic use ; Antiviral Agents/chemistry ; Enfuvirtide/therapeutic use ; Peptides/pharmacology ; Peptides/chemistry
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