Suchergebnisse - "Aconitine analogs & derivatives"

[3H]A-585539 [(1 S,4 S)-2,2-Dimethyl-5-(6-phenylpyridazin-3-yl)-5-aza-2-azoniabicyclo[2.2.1]heptane], a Novel High-Affinity α7 Neuronal Nicotinic Receptor Agonist: Radioligand Binding Characterization to Rat and Human Brain

Autoren: Anderson, David J. Bunnelle, William Surber, Bruce et al.

Quelle: Journal of Pharmacology and Experimental Therapeutics, Vol. 324, No 1 (2008) pp. 179-187

Schlagwörter: Aconitine/analogs & derivatives/metabolism, Bridged-Ring Compounds, Nicotine, 616.8, alpha7 Nicotinic Acetylcholine Receptor, Aconitine, Nicotinic Antagonists, Receptors, Nicotinic, Cell Line, Rats, Sprague-Dawley, Bridged Bicyclo Compounds, Radioligand Assay, 03 medical and health sciences, 0302 clinical medicine, Receptors, Nicotinic/*metabolism, Nicotinic Agonists/*metabolism, Benzamides/metabolism, Animals, Humans, Spiro Compounds, Nicotinic Agonists, Nicotinic Antagonists/metabolism, Bungarotoxins/metabolism, Pyridazines/*metabolism, Spiro Compounds/metabolism, Brain, Bicyclo Compounds/metabolism, Bridged Bicyclo Compounds, Heterocyclic, Bungarotoxins, ddc:616.8, Bicyclo Compounds, Heterocyclic/*metabolism, Rats, Pyridazines, Benzamides, Bridged Compounds/metabolism, Nicotine/metabolism, Brain/*metabolism

Dateibeschreibung: application/pdf

Zugangs-URL: https://pubmed.ncbi.nlm.nih.gov/17959745
http://jpet.aspetjournals.org/content/jpet/324/1/179.full.pdf
https://www.ncbi.nlm.nih.gov/pubmed/17959745
https://jpet.aspetjournals.org/content/324/1/179
http://europepmc.org/abstract/MED/17959745
http://jpet.aspetjournals.org/content/early/2007/10/24/jpet.107.130062.full.pdf
https://archive-ouverte.unige.ch/unige:19154
https://archive-ouverte.unige.ch/unige:19154
https://archive-ouverte.unige.ch/unige:19154
https://doi.org/10.1124/jpet.107.130062

Inhibition of both α7* and β2* nicotinic acetylcholine receptors is necessary to prevent development of sensitization to cocaine-elicited increases in extracellular dopamine levels in the ventral striatum

Autoren: Lara Zanetti Alban de Kerchove d'Exaerde Jean-Pierre Changeux et al.

Weitere Verfasser: Lara Zanetti Alban de Kerchove d'Exaerde Jean-Pierre Changeux et al.

Quelle: Psychopharmacology. 187:181-188

Schlagwörter: Male, alpha7 Nicotinic Acetylcholine Receptor, Knockout, Aconitine, Dopamine, Nicotinic Antagonists, Mecamylamine, Receptors, Nicotinic, Inbred C57BL, Basal Ganglia, Nicotinic -- drug effects, Mice, 03 medical and health sciences, 0302 clinical medicine, Aconitine -- analogs & derivatives, Cocaine, Cocaine -- pharmacology, Receptors, Animals, Nicotinic Antagonists -- pharmacology, Aconitine -- pharmacology, Basal Ganglia -- drug effects, Central Nervous System Stimulants -- pharmacology, Mecamylamine -- pharmacology, Mice, Knockout, Extracellular Fluid -- drug effects, [SDV.NEU.NB] Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]/Neurobiology, cocaine, dopamine, mecamylamine, methyllycaconitine, microdialysis, mice, knockout, Extracellular Fluid, Sciences bio-médicales et agricoles, 3. Good health, Mice, Inbred C57BL, Dopamine -- metabolism, Central Nervous System Stimulants

Dateibeschreibung: 1 full-text file(s): application/pdf

Zugangs-URL: https://pubmed.ncbi.nlm.nih.gov/16826402
https://pasteur.hal.science/pasteur-00161386v1
https://doi.org/10.1007/s00213-006-0419-y
https://iris.unimore.it/handle/11380/304909
https://difusion.ulb.ac.be/vufind/Record/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/50715/Details
https://link.springer.com/article/10.1007%2Fs00213-006-0419-y
https://pubmed.ncbi.nlm.nih.gov/16826402/
https://iris.univr.it/handle/11562/313250
https://link.springer.com/content/pdf/10.1007%2Fs00213-006-0419-y.pdf
https://hdl.handle.net/11562/313250
https://hdl.handle.net/11380/304909
https://doi.org/10.1007/s00213-006-0419-y

Identified spinal motoneurons of young rats possess nicotinic acetylcholine receptors of the heteromeric family

Autoren: Ogier, R. Liu, X. Tribollet, Eliane et al.

Quelle: European Journal of Neuroscience, Vol. 20, No 10 (2004) pp. 2591-2597

Schlagwörter: 0301 basic medicine, 616.8, Patch-Clamp Techniques, Patch-Clamp Techniques/methods, Iodine Isotopes/pharmacokinetics, Aconitine, Pyridines/pharmacokinetics/pharmacology, Autoradiography/methods, Nicotinic Antagonists, Bungarotoxins/pharmacokinetics, In Vitro Techniques, Tritium/pharmacokinetics, Choline O-Acetyltransferase, Membrane Potentials, Nicotinic Antagonists/pharmacology, Rats, Sprague-Dawley, Spinal Cord/ cytology, 03 medical and health sciences, 0302 clinical medicine, Choline O-Acetyltransferase/metabolism, Iodine Isotopes, Immunohistochemistry/methods, Animals, Lysine/ analogs & derivatives/metabolism, Nicotinic Agonists, Tubocurarine/pharmacology, Motor Neurons, Acetylcholine/pharmacology, Binding Sites, Lysine, Motor Neurons/drug effects/ metabolism, Age Factors, Dihydro-beta-Erythroidine, Bridged Bicyclo Compounds, Heterocyclic, Bungarotoxins, Immunohistochemistry, Acetylcholine, ddc:616.8, Rats, Bicyclo Compounds, Heterocyclic/pharmacokinetics/pharmacology, Animals, Newborn, Receptors, Nicotinic/classification/drug effects/ metabolism, Autoradiography, Aconitine/ analogs & derivatives/pharmacology, Dihydro-beta-Erythroidine/pharmacology, Membrane Potentials/drug effects/physiology, Nicotinic Agonists/pharmacokinetics

Dateibeschreibung: application/pdf

Zugangs-URL: https://pubmed.ncbi.nlm.nih.gov/15548202
https://core.ac.uk/display/60772103
https://onlinelibrary.wiley.com/doi/10.1111/j.1460-9568.2004.03746.x
https://archive-ouverte.unige.ch/unige:10379
https://pubmed.ncbi.nlm.nih.gov/15548202/
https://www.ncbi.nlm.nih.gov/pubmed/15548202
https://archive-ouverte.unige.ch/unige:10379

Modulation of synaptic transmission by nicotine and nicotinic antagonists in hippocampus

Autoren: Chiodini, F. C. Tassonyi, Edomer Hulo, S. et al.

Quelle: Brain Research Bulletin, Vol. 48, No 6 (1999) pp. 623-628

Schlagwörter: Nicotine, 616.8, Nicotine/ pharmacology, Aconitine, Neural Inhibition/drug effects/physiology, Nicotinic Antagonists, In Vitro Techniques, Mecamylamine, Hippocampus, Synaptic Transmission, Rats, Sprague-Dawley, 03 medical and health sciences, Nicotinic Antagonists/ pharmacology, 0302 clinical medicine, Mecamylamine/pharmacology, Animals, Hippocampus/ drug effects/ physiology, Neural Inhibition, Dihydro-beta-Erythroidine, ddc:616.8, Rats, 3. Good health, Synaptic Transmission/ drug effects, Aconitine/analogs & derivatives/pharmacology, Dihydro-beta-Erythroidine/pharmacology

Dateibeschreibung: application/pdf

Zugangs-URL: https://pubmed.ncbi.nlm.nih.gov/10386843
https://www.ncbi.nlm.nih.gov/pubmed/10386843
https://archive-ouverte.unige.ch/unige:10215
https://europepmc.org/abstract/MED/10386843
https://pubmed.ncbi.nlm.nih.gov/10386843/
https://www.sciencedirect.com/science/article/pii/S036192309900043X
https://archive-ouverte.unige.ch/unige:10215

Synaptic transmission at nicotinic acetylcholine receptors in rat hippocampal organotypic cultures and slices

Autoren: Hefft, S. Hulo, S. Bertrand, Daniel et al.

Quelle: The Journal of Physiology, Vol. 515 ( Pt 3) (1999) pp. 769-776

Schlagwörter: 616.8, Synaptic Transmission/drug effects/ physiology, Aconitine, Tubocurarine, Nicotinic Antagonists, Pyramidal Cells/drug effects/ physiology, Receptors, Nicotinic, Excitatory Amino Acid Antagonists/ pharmacology, Hippocampus, Synaptic Transmission, Bungarotoxins/pharmacology, Piperazines, Nicotinic Antagonists/pharmacology, GABA Antagonists, Rats, Sprague-Dawley, 03 medical and health sciences, Organ Culture Techniques, 0302 clinical medicine, Picrotoxin/pharmacology, Quinoxalines, Animals, Picrotoxin, Piperazines/pharmacology, Evoked Potentials, Tubocurarine/pharmacology, Pyramidal Cells, Receptors, Nicotinic/ physiology, Bungarotoxins, ddc:616.8, Quinoxalines/pharmacology, Rats, GABA Antagonists/pharmacology, Evoked Potentials/drug effects, Aconitine/analogs & derivatives/pharmacology, Hippocampus/ physiology, Excitatory Amino Acid Antagonists

Dateibeschreibung: application/pdf

Zugangs-URL: https://physoc.onlinelibrary.wiley.com/doi/pdfdirect/10.1111/j.1469-7793.1999.769ab.x
https://pubmed.ncbi.nlm.nih.gov/10066903
https://physoc.onlinelibrary.wiley.com/doi/10.1111/j.1469-7793.1999.769ab.x
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2269188/
http://europepmc.org/abstract/MED/10066903
https://archive-ouverte.unige.ch/unige:10296
https://stemcellsjournals.onlinelibrary.wiley.com/doi/10.1111/j.1469-7793.1999.769ab.x
http://onlinelibrary.wiley.com/doi/10.1111/j.1469-7793.1999.769ab.x/full
https://archive-ouverte.unige.ch/unige:10296

Agonist actions of clothianidin on synaptic and extrasynaptic nicotinic acetylcholine receptors expressed on cockroach sixth abdominal ganglion

Autoren: S.H. Thany

Quelle: Neurotoxicology

Schlagwörter: Acetylcholine/pharmacology, Aconitine/analogs & derivatives/pharmacology, Analysis of Variance, Animals, Biophysics, Cockroaches, Dose-Response Relationship, Drug, Electric Stimulation, Excitatory Postsynaptic Potentials/drug effects, Ganglia, Invertebrate/cytology/drug effects, Gene Expression Regulation/drug effects, Guanidines/pharmacology, Male, Neurons/drug effects, Nicotine/pharmacology, Nicotinic Agonists/pharmacology, Nicotinic Antagonists/pharmacology, Patch-Clamp Techniques, Receptors, Nicotinic/genetics/metabolism, Synapses/drug effects, Thiazoles/pharmacology

Relation: http://okina.univ-angers.fr/publications/ua7539

Verfügbarkeit: http://okina.univ-angers.fr/publications/ua7539
https://doi.org/10.1016/j.neuro.2009.06.013

[3H]A-585539 [(1S,4S)-2,2-dimethyl-5-(6-phenylpyridazin-3-yl)-5-aza-2-azoniabicyclo[2.2 .1]heptane], a novel high-affinity alpha7 neuronal nicotinic receptor agonist: radioligand binding characterization to rat and human brain

Autoren: Anderson, David J. Bunnelle, William Surber, Bruce et al.

Quelle: ISSN: 0022-3565 ; The Journal of pharmacology and experimental therapeutics, vol. 324, no. 1 (2008) p. 179-187.

Schlagwörter: info:eu-repo/classification/ddc/616.8, Aconitine/analogs & derivatives/metabolism, Animals, Benzamides/metabolism, Bicyclo Compounds/metabolism, Bicyclo Compounds, Heterocyclic/*metabolism, Brain/*metabolism, Bridged Compounds/metabolism, Bungarotoxins/metabolism, Cell Line, Humans, Nicotine/metabolism, Nicotinic Agonists/*metabolism, Nicotinic Antagonists/metabolism, Pyridazines/*metabolism, Radioligand Assay, Rats, Sprague-Dawley, Receptors, Nicotinic/*metabolism, Spiro Compounds/metabolism

Relation: info:eu-repo/semantics/altIdentifier/pmid/17959745; unige:19154

Verfügbarkeit: https://archive-ouverte.unige.ch/unige:19154

Inhibition of both alpha7* and beta2* nicotinic acetylcholine receptors is necessary to prevent development of sensitization to cocaine-elicited increases in extracellular dopamine levels in the ventral striatum.

Autoren: Zanetti, Lara de Kerchove d'Exaerde, Alban Zanardi, Alessio et al.

Quelle: Psychopharmacologia, 187 (2

Schlagwörter: Sciences bio-médicales et agricoles, Aconitine -- analogs & derivatives, Aconitine -- pharmacology, Animals, Basal Ganglia -- drug effects, Central Nervous System Stimulants -- pharmacology, Cocaine -- pharmacology, Dopamine -- metabolism, Extracellular Fluid -- drug effects, Male, Mecamylamine -- pharmacology, Mice, Inbred C57BL, Knockout, Nicotinic Antagonists -- pharmacology, Receptors, Nicotinic -- drug effects

Dateibeschreibung: 1 full-text file(s): application/pdf

Relation: uri/info:pmid/16826402; uri/info:scp/33745751083; https://dipot.ulb.ac.be/dspace/bitstream/2013/50715/1/Psychopharmacology2006Zanetti.pdf

Verfügbarkeit: https://hdl.handle.net/2013/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/50715
https://dipot.ulb.ac.be/dspace/bitstream/2013/50715/1/Psychopharmacology2006Zanetti.pdf